Posaconazole 171228-49-2 Tshuaj tua kab mob
Kev Them Nyiaj:T / T, L / C
Khoom Keeb Kwm:Tuam Tshoj
Shipping Chaw nres nkoj:Beijing / Shanghai / Hangzhou
Muaj peev xwm ntau lawm:20kg / hli
Order (MOQ):10g ua
Lub Sijhawm Lead:3 Hnub Ua Haujlwm
Kev cia khoom:Khaws rau hauv qhov chaw txias, qhuav, chav sov.
Cov khoom siv pob:vial
Pob loj:10g / vial
Cov ntaub ntawv kev nyab xeeb:Tsis yog khoom txaus ntshai

Taw qhia
Posaconazole yog tshuaj tua kab mob triazole.
Posaconazole yog siv los kho cov kab mob Aspergillus thiab Candida invasive.Nws kuj tseem siv rau kev kho mob ntawm oropharyngeal candidiasis (OPC), suav nrog OPC refractory rau itraconzaole thiab / lossis fluconazole therapy.
Nws kuj tseem siv los kho cov kab mob kis los ntawm Candida, Mucor, thiab Aspergillus hom kab mob hauv cov neeg mob hnyav.
Specification (hauv tsev qauv)
Yam khoom | Specification |
Qhov tshwm sim | Dawb los yog yuav luag dawb, hygroscopic hmoov |
Yam khoom | Specification |
Qhov tshwm sim | Dawb los yog tawm-dawb crystalline hmoov |
Kev sib hloov tshwj xeeb | -28.0° ~ 34.0° |
Crystal daim ntawv | Nws yuav tsum yog crystalline Ⅰ, nrog 2-theta kaum ntawm 14.4 ± 0.2 °, 19.2 ± 0.2 °, 21.7 ± 0.2 °, 24.3 ± 0.2 ° 29.3 ± 0.2 ° |
Kev txheeb xyuas | IR, HPLC |
Cov khoom muaj feem xyuam I | PO-R1 NMT 0.10% |
PO-R2 NMT 0.10% | |
PO-R3 NMT 0.10% | |
PO-R4 NMT 0.10% | |
PO-D3 & PO-D5 NMT 0.10% | |
PO-D7 & PO-D10 NMT 0.10% | |
Txhua yam ntawm impurity NMT 0.10% | |
Tag nrho impurities NMT 0.5% | |
Cov khoom muaj feem cuam tshuam Ⅱ | PO-E NMT 0.10% |
PO-D1 NMT 0.10% | |
PO-R5 NMT 0.10% | |
Cov kuab tshuaj residual | Methanol NMT 3000ppm |
Ethanol NMT 5000ppm | |
Tom ntej: Dichloromethane NMT 600ppm | |
Tom ntej: Tetrahydrofuran NMT 720ppm | |
N, N-dimethylformamide NMT 880ppm | |
Tom ntej: Triethylamine NMT 100ppm | |
Dimethy sulfoxide NMT 5000ppm | |
Dej | 2.0% NMT |
Residue ntawm ignition | NMT 0.1% |
Cov hlau hnyav | NMT 10 ppm |
Microbial txwv | Tag nrho aerobic NMT 1000cfu / g Tag nrho cov poov xab thiab pwm NMT 100cfu / g E.coli yuav tsum tsis tuaj |
Assay | 98.0% -102.0% (raws li anhydrous hauv paus) |
98.0% -102.0% (ntawm anhydrous thiab solvents dawb hauv paus) |